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Number of items: 2.
2019
Sijm, Maarten and Siciliano de Araújo, Julianna and Kunz, Stefan and Schroeder, Susanne and Edink, Ewald and Orrling, Kristina M. and Matheeussen, An and van de Meer, Tiffany and Sadek, Payman and Custers, Hans and Cotillo, Ignacio and Martin, Julio J. and Siderius, Marco and Maes, Louis and Brown, David G. and de Nazaré Correia Soeiro, Maria and Sterk, GeertJan and de Esch, Iwan J.P. and Leurs, Rob (2019) Phenyldihydropyrazolones as Novel Lead Compounds Against Trypanosoma cruzi. ACS Omega, 4 (4). pp. 6585-6596. ISSN 2470-1343. (doi:https://doi.org/10.1021/acsomega.8b02847) (Full text available) |
2018
Blaazer, Antoni R. and Singh, Abhimanyu K. and de Heuvel, Erik and Edink, Ewald and Orrling, Kristina M. and Veerman, Johan J. N. and van den Bergh, Toine and Jansen, Chimed and Balasubramaniam, Erin and Mooij, Wouter J. and Custers, Hans and Sijm, Maarten and Tagoe, Daniel N. A. and Kalejaiye, Titilola D. and Munday, Jane C. and Tenor, Hermann and Matheeussen, An and Wijtmans, Maikel and Siderius, Marco and de Graaf, Chris and Maes, Louis and de Koning, Harry P. and Bailey, David S. and Sterk, Geert Jan and de Esch, Iwan J. P. and Brown, David G. and Leurs, Rob (2018) Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity. Journal of Medicinal Chemistry, 61 (9). pp. 3870-3888. ISSN 0022-2623. (doi:https://doi.org/10.1021/acs.jmedchem.7b01670) (Full text available) |